AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2

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Authors: Frank Narjes, Antonio Llinas, Stefan von Berg, Johan Jirholt, Sarah Lever, Rikard Pehrson, Mia Collins, Anna Malmberg, Petter Svanberg, Yafeng Xue, Roine I. Olsson, Jesper Malmberg, Glyn Hughes, Nafizal Hossain, Hanna Grindebacke, Agnes Leffler, Nina Krutrök, Elisabeth Bäck, Marie Ramnegård, Matti Lepistö, Linda Thunberg, Anna Aagaard, Jane McPheat, Eva L. Hansson, Rongfeng Chen, Yao Xiong, Thomas G. Hansson

J Med Chem. 2021 Sep 23;64(18):13807-13829

DOI: 10.1021/acs.jmedchem.1c01197

Access the publication at:https://pubmed.ncbi.nlm.nih.gov/34464130/