Discovery of AZD8154, a dual PI3Kγδ inhibitor for the treatment of asthma

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Authors: Matthew W. D. Perry, Karin Björhall, Peter Bold, Mikael Brűlls, Ulf Börjesson, Johan Carlsson, Hui-Fang Amy Chang, Yunhua Chen, Anders Eriksson, Britt-Marie Fihn, Rebecca Fransson, Linda Fredlund, Hongbin Ge, Haijuan Huang, Kostas Karabelas, Eva Lamm Bergström, Sarah Lever, Helena Lindmark, Mickael Mogemark, Antonios Nikitidis, Anna-Pia Palmgren, Nils Pemberton, Jens Petersen, Mio Rodrigo Blomqvist, Reed W. Smith, Matthew J. Thomas , Victoria Ullah, Christian Tyrchan, Tiiu Wennberg, Annika Westin Eriksson, Wenzhen Yang, Shuchun Zhao, Linda Öster
J Med Chem. 2021 Jun 24;64(12):8053-8075
DOI: 10.1021/acs.jmedchem.1c00434
Access the publication at:https://pubmed.ncbi.nlm.nih.gov/34080862/