Structure-guided design of a selective inhibitor of the methyltransferase KMT9 with cellular activity

Capabilities
Authors: Sheng Wang, Sebastian O. Klein, Sylvia Urban, Maximilian Staudt, Nicolas P. F. Barthes, Dominica Willmann, Johannes Bacher, Manuela Sum, Helena Bauer, Ling Peng, Georg A. Rennar, Christian Gratzke, Katrin M. Schüle, Lin Zhang, Oliver Einsle, Holger Greschik, Calum MacLeod, Christopher G. Thomson, Manfred Jung, Eric Metzger, Roland Schüle
Nat Commun. 2024 Jan 2;15(1):43
DOI: 10.1038/s41467-023-44243-6
Access the publication at:https://pubmed.ncbi.nlm.nih.gov/38167811/