Structure-guided design of novel, potent, and selective macrocyclic plasma kallikrein inhibitors

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Authors: Zhe Li, James Partridge, Abel Silva-Garcia, Peter Rademacher, Andreas Betz, Qing Xu, Hing Sham, Yunjin Hu, Yuqing Shan, Bin Liu, Ying Zhang, Haijuan Shi, Qiong Xu, Xubo Ma, Li Zhang
ACS Med Chem Lett. 2016 Dec 6;8(2):185-190
DOI: 10.1021/acsmedchemlett.6b00384
Access the publication at:https://pubmed.ncbi.nlm.nih.gov/28197309/