Publications

Publications

On-DNA Morita-Baylis-Hillman Reaction: Accessing Targeted Covalent Inhibitor Motifs in DNA-Encoded Libraries

Xue, L.; Liu, W.; Li, S.; Duchemin, N.; Lou, M.; Yuan, J.; Zhang, H.; Chen, J.; Yu, W.; Yang, K.; Hu, Y.J. Bioconjugate Chem., 2023.
Publications

Develpment of On-DNA Thiophene Synthesis for DEL Construction

Luo, A.; Duchemin, N.; Wang, X.; Zhou, H.; Zeng, F.; Zhao, X.; Yu, W.; Yang, K.; Hu, Y.J. Chemistry: An Asian Journal. 2023. (Link)
Publications

Constructive on-DNA Thiol Aerial Oxidization for DNA-encoded Library Synthesis

Sun, Z.; Xiao, L.; Chen, Y.; Wang, J.; Zeng, F.; Zhang, H.; Zhang, J.; Yang, K.; Hu, Y.J. ACS Med. Chem. Lett. 2023, 14, 4, 473-478.
Publications

Development of the Inverse Sonogashira Reaction for DEL Synthesis

Luo, A.; Zhou, H.; Hua, Q.; An, Y.; Ma, H.; Zhao, X.; Yang, K.; Hu, Y.J., ACS Med. Chem. Lett. 2023, 14, 3, 270-277.
Publications

On-DNA Alkyne Iodination and Acetylenic Coupling as a Useful Tool for DEL Synthesis

Ayun, L.; Zhou, H.; Zhou, Q.; Hua, Q.; Zhao, X.; Yu, X.; Yang, K.; Hu, Y.J., Bioconjugate Chem., 2022, 33, 12, 2299-2306.